Sfoglia per Autore RADI, MARCO
Studies on the ATP Binding Site of Fyn Kinase for the Identification of New Inhibitors and Their Evaluation as Potential Agents against Tauopathies and Tumors
2015-01-01 Tintori, Cristina; La Sala, Giuseppina; Vignaroli, Giulia; Botta, Lorenzo; Fallacara, Anna Lucia; Falchi, Federico; Radi, Marco; Zamperini, Claudio; Dreassi, Elena; Dello Iacono, Lucia; Orioli, Donata; Biamonti, Giuseppe; Garbelli, Mirko; Lossani, Andrea; Gasparrini, Francesca; Tuccinardi, Tiziano; Laurenzana, Ilaria; Angelucci, Adriano; Maga, Giovanni; Schenone, Silvia; Brullo, Chiara; Musumeci, Francesca; Desogus, Andrea; Crespan, Emmanuele; Botta, Maurizio
Combining X-ray Crystallography and Molecular Modeling toward the Optimization of Pyrazolo[3,4-d]pyrimidines as Potent c-Src Inhibitors Active in Vivo against Neuroblastoma
2015-01-01 Tintori, Cristina; Fallacara, A. L.; Radi, Marco; Zamperini, Claudio; Dreassi, Elena; Crespan, E.; Maga, G.; Schenone, S.; Musumeci, F.; Brullo, C.; Richters, A.; Gasparrini, F.; Angelucci, A.; Festuccia, C.; Delle Monache, S.; Rauh, D.; Botta, M.
CYP-dependent metabolism of antitumor pyrazolo[3,4-d]pyrimidine derivatives is characterized by an oxidative dechlorination reaction
2014-01-01 Zamperini, C.; Dreassi, E.; Vignaroli, G.; Radi, M.; Dragoni, S.; Schenone, S.; Musumeci, F.; Valoti, M.; Antiochia, R.; Botta, M.
Pyrazolo[3,4-d]pyrimidine Prodrugs: Strategic Optimization of the Aqueous Solubility of Dual Src/Abl Inhibitors
2013-01-01 Vignaroli, Giulia; Zamperini, Claudio; Dreassi, Elena; Radi, Marco; Angelucci, A.; Sanità, P.; Crespan, E.; Kissova, M.; Maga, G.; Schenone, S.; Musumeci, F.; Botta, Maurizio
A combined targeted/phenotypic approach for the identification of new antiangiogenics agents active on a zebrafish model:from in silico screening to cyclodextrin formulation
2012-01-01 Radi, M.; Evensen, L.; Dreassi, E.; Zamperini, C.; Caporicci, M.; Falchi, F.; Musumeci, A.; Schenone, S.; Lorens, J. B.; Botta, M.
Targeting the human DEAD-box polypeptide 3 (DDX3) RNA helicase as a novel strategy to inhibit viral replication
2011-01-01 Garbelli, A.; Radi, M.; Falchi, F.; Beermann, S.; Zanoli, S.; Manetti, F.; Dietrich, U.; Botta, M.; Maga, G.
Design, synthesis, biological activity and ADME properties of pyrazolo[3,4-d]pyrimidines active in hypoxic human leukemia cells: a lead optimization study
2011-01-01 Radi, Marco; Dreassi, Elena; C., Brullo; E., Crespan; Tintori, Cristina; V., Bernardo; Valoti, Massimo; Zamperini, Claudio; H., Daigl; F., Musumeci; Carraro, Fabio; Naldini, Antonella; Filippi, Irene; G., Maga; S., Schenone; Botta, Maurizio
New insights into small-molecule inhibitors of Bcr-Abl
2010-01-01 Schenone, S.; Botta, Maurizio; Radi, Marco; Bruno, O.
A Practical One-Pot Two-Step Protocol for the Microwave-Assisted Synthesis of Highly Functionalized Rhodanine Derivatives
2010-01-01 Radi, Marco; Botta, Lorenzo; Casaluce, Gianni; Bernardini, Martina; Botta, Maurizio
Crystal Structure of HIV-1 Reverse Transcriptase Bound to a Non-Nucleoside Inhibitor with a Novel Mechanism of Action
2010-01-01 Freisz, S.; Bec, G.; Radi, Marco; Wolff, P.; Crespan, E.; Angeli, Lucilla; Dumas, P.; Maga, G.; Botta, Maurizio; Ennifar, E.
HIV-1 RT inhibitors with a novel mechanism of action: NNRTIs that compete with the nucleotide substrate
2010-01-01 Maga, G.; Radi, Marco; Gerard, M.; Botta, Maurizio; Ennifar, E.
Arylation of 2-Furyl 4-Fluorophenyl Ketone: an extension of Heck Chemistry towards Novel Integrase Inhibitors
2010-01-01 Franchi, Luigi; Rinaldi, Marta; Vignaroli, Giulia; Innitzer, Anna; Radi, Marco; Botta, Maurizio
NEW 4-SUBSTITUTED DERIVATIVES OF PYRAZOLO[3,4-D PYRIMIDINE AND PYRROLO[2,3-D]PYRIMIDINE AND USES THEREOF | [NOUVEAUX DÉRIVÉS 4-SUBSTITUÉS DE LA PYRAZOLO[3,4-D]PYRIMIDINE ET DE LA PYRROLO[2,3-D]PYRIMIDINE ET LEURS UTILISATIONS]
2009-01-01 Schenone, Silvia; Bondavalli, Francesco; Bruno, Olga; Botta, Maurizio; Manetti, Fabrizio; Radi, Marco; Santucci, Alessandra; Maga, Giovanni; Bologna, Mauro; Angelucci, Adriano; Santucci, Annalisa; Spreafico, Adriano; Carraro, Fabio; Borlak, Jurgen
Microwave-assisted organocatalytic multicomponent Knoevenagel/Hetero Diels Alder reaction for the synthesis of 2,3-dihydropyran[2,3-c]pyrazoles
2009-01-01 Radi, Marco; Bernardo, Vincenzo; Bechi, Beatrice; Castagnolo, Daniele; Pagano, Mafalda; Botta, Maurizio
Recent highlights in the synthesis of highly functionalized pyrimidines
2009-01-01 Radi, Marco; Botta, Maurizio; Schenone, S.
4-Aminosubstituted pyrazolo[3,4d]pyrimidines: synthesis and biological properties
2009-01-01 Schenone, S.; Bruno, O.; Radi, Marco; Botta, Maurizio
A Multidisciplinary Approach for the Identification ofNovel HIV-1 Non-Nucleoside Reverse TranscriptaseInhibitors: S-DABOCs and DAVPs
2008-01-01 Radi, Marco; Falciani, Chiara; Contemori, Lorenzo; Petricci, Elena; Maga, G.; Samuele, A.; Zanoli, S.; Terrazas, M.; Castria, Marinunzia; Togninelli, Andrea; Esté, J. A.; Clotet Codina, I.; Armand Ugon, M.; Botta, Maurizio
A one-pot, two step microwave-assisted synthesis of highly functionalized benzoxazoles using solid-supported reagents (SSRs)
2008-01-01 Radi, Marco; Saletti, S.; Botta, Maurizio
6-Vinyl pyrimidine and pyrimidinone derivatives and the use thereof
2007-01-01 Botta, Maurizio; Corelli, Federico; Petricci, Elena; Radi, Marco; Giovanni, Maga; JOSE A., Este; Antonello, Mai
Microwave-enhanced Sonogashira coupling reaction of substituted pyrimidinones and pyrimidine nucleosides
2003-01-01 Petricci, Elena; Radi, Marco; Corelli, Federico; Botta, Maurizio
Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
---|---|---|---|---|
Studies on the ATP Binding Site of Fyn Kinase for the Identification of New Inhibitors and Their Evaluation as Potential Agents against Tauopathies and Tumors | 1-gen-2015 | Tintori, Cristina; La Sala, Giuseppina; Vignaroli, Giulia; Botta, Lorenzo; Fallacara, Anna Lucia; Falchi, Federico; Radi, Marco; Zamperini, Claudio; Dreassi, Elena; Dello Iacono, Lucia; Orioli, Donata; Biamonti, Giuseppe; Garbelli, Mirko; Lossani, Andrea; Gasparrini, Francesca; Tuccinardi, Tiziano; Laurenzana, Ilaria; Angelucci, Adriano; Maga, Giovanni; Schenone, Silvia; Brullo, Chiara; Musumeci, Francesca; Desogus, Andrea; Crespan, Emmanuele; Botta, Maurizio | - | |
Combining X-ray Crystallography and Molecular Modeling toward the Optimization of Pyrazolo[3,4-d]pyrimidines as Potent c-Src Inhibitors Active in Vivo against Neuroblastoma | 1-gen-2015 | Tintori, Cristina; Fallacara, A. L.; Radi, Marco; Zamperini, Claudio; Dreassi, Elena; Crespan, E.; Maga, G.; Schenone, S.; Musumeci, F.; Brullo, C.; Richters, A.; Gasparrini, F.; Angelucci, A.; Festuccia, C.; Delle Monache, S.; Rauh, D.; Botta, M. | - | |
CYP-dependent metabolism of antitumor pyrazolo[3,4-d]pyrimidine derivatives is characterized by an oxidative dechlorination reaction | 1-gen-2014 | Zamperini, C.; Dreassi, E.; Vignaroli, G.; Radi, M.; Dragoni, S.; Schenone, S.; Musumeci, F.; Valoti, M.; Antiochia, R.; Botta, M. | - | |
Pyrazolo[3,4-d]pyrimidine Prodrugs: Strategic Optimization of the Aqueous Solubility of Dual Src/Abl Inhibitors | 1-gen-2013 | Vignaroli, Giulia; Zamperini, Claudio; Dreassi, Elena; Radi, Marco; Angelucci, A.; Sanità, P.; Crespan, E.; Kissova, M.; Maga, G.; Schenone, S.; Musumeci, F.; Botta, Maurizio | - | |
A combined targeted/phenotypic approach for the identification of new antiangiogenics agents active on a zebrafish model:from in silico screening to cyclodextrin formulation | 1-gen-2012 | Radi, M.; Evensen, L.; Dreassi, E.; Zamperini, C.; Caporicci, M.; Falchi, F.; Musumeci, A.; Schenone, S.; Lorens, J. B.; Botta, M. | - | |
Targeting the human DEAD-box polypeptide 3 (DDX3) RNA helicase as a novel strategy to inhibit viral replication | 1-gen-2011 | Garbelli, A.; Radi, M.; Falchi, F.; Beermann, S.; Zanoli, S.; Manetti, F.; Dietrich, U.; Botta, M.; Maga, G. | - | |
Design, synthesis, biological activity and ADME properties of pyrazolo[3,4-d]pyrimidines active in hypoxic human leukemia cells: a lead optimization study | 1-gen-2011 | Radi, Marco; Dreassi, Elena; C., Brullo; E., Crespan; Tintori, Cristina; V., Bernardo; Valoti, Massimo; Zamperini, Claudio; H., Daigl; F., Musumeci; Carraro, Fabio; Naldini, Antonella; Filippi, Irene; G., Maga; S., Schenone; Botta, Maurizio | - | |
New insights into small-molecule inhibitors of Bcr-Abl | 1-gen-2010 | Schenone, S.; Botta, Maurizio; Radi, Marco; Bruno, O. | - | |
A Practical One-Pot Two-Step Protocol for the Microwave-Assisted Synthesis of Highly Functionalized Rhodanine Derivatives | 1-gen-2010 | Radi, Marco; Botta, Lorenzo; Casaluce, Gianni; Bernardini, Martina; Botta, Maurizio | - | |
Crystal Structure of HIV-1 Reverse Transcriptase Bound to a Non-Nucleoside Inhibitor with a Novel Mechanism of Action | 1-gen-2010 | Freisz, S.; Bec, G.; Radi, Marco; Wolff, P.; Crespan, E.; Angeli, Lucilla; Dumas, P.; Maga, G.; Botta, Maurizio; Ennifar, E. | - | |
HIV-1 RT inhibitors with a novel mechanism of action: NNRTIs that compete with the nucleotide substrate | 1-gen-2010 | Maga, G.; Radi, Marco; Gerard, M.; Botta, Maurizio; Ennifar, E. | - | |
Arylation of 2-Furyl 4-Fluorophenyl Ketone: an extension of Heck Chemistry towards Novel Integrase Inhibitors | 1-gen-2010 | Franchi, Luigi; Rinaldi, Marta; Vignaroli, Giulia; Innitzer, Anna; Radi, Marco; Botta, Maurizio | - | |
NEW 4-SUBSTITUTED DERIVATIVES OF PYRAZOLO[3,4-D PYRIMIDINE AND PYRROLO[2,3-D]PYRIMIDINE AND USES THEREOF | [NOUVEAUX DÉRIVÉS 4-SUBSTITUÉS DE LA PYRAZOLO[3,4-D]PYRIMIDINE ET DE LA PYRROLO[2,3-D]PYRIMIDINE ET LEURS UTILISATIONS] | 1-gen-2009 | Schenone, Silvia; Bondavalli, Francesco; Bruno, Olga; Botta, Maurizio; Manetti, Fabrizio; Radi, Marco; Santucci, Alessandra; Maga, Giovanni; Bologna, Mauro; Angelucci, Adriano; Santucci, Annalisa; Spreafico, Adriano; Carraro, Fabio; Borlak, Jurgen | - | |
Microwave-assisted organocatalytic multicomponent Knoevenagel/Hetero Diels Alder reaction for the synthesis of 2,3-dihydropyran[2,3-c]pyrazoles | 1-gen-2009 | Radi, Marco; Bernardo, Vincenzo; Bechi, Beatrice; Castagnolo, Daniele; Pagano, Mafalda; Botta, Maurizio | - | |
Recent highlights in the synthesis of highly functionalized pyrimidines | 1-gen-2009 | Radi, Marco; Botta, Maurizio; Schenone, S. | - | |
4-Aminosubstituted pyrazolo[3,4d]pyrimidines: synthesis and biological properties | 1-gen-2009 | Schenone, S.; Bruno, O.; Radi, Marco; Botta, Maurizio | - | |
A Multidisciplinary Approach for the Identification ofNovel HIV-1 Non-Nucleoside Reverse TranscriptaseInhibitors: S-DABOCs and DAVPs | 1-gen-2008 | Radi, Marco; Falciani, Chiara; Contemori, Lorenzo; Petricci, Elena; Maga, G.; Samuele, A.; Zanoli, S.; Terrazas, M.; Castria, Marinunzia; Togninelli, Andrea; Esté, J. A.; Clotet Codina, I.; Armand Ugon, M.; Botta, Maurizio | - | |
A one-pot, two step microwave-assisted synthesis of highly functionalized benzoxazoles using solid-supported reagents (SSRs) | 1-gen-2008 | Radi, Marco; Saletti, S.; Botta, Maurizio | - | |
6-Vinyl pyrimidine and pyrimidinone derivatives and the use thereof | 1-gen-2007 | Botta, Maurizio; Corelli, Federico; Petricci, Elena; Radi, Marco; Giovanni, Maga; JOSE A., Este; Antonello, Mai | - | |
Microwave-enhanced Sonogashira coupling reaction of substituted pyrimidinones and pyrimidine nucleosides | 1-gen-2003 | Petricci, Elena; Radi, Marco; Corelli, Federico; Botta, Maurizio | - |
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